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Table 1 Isolated yields of amide 2, sulfonamide 3 and urea 4 derivatives

From: Sucrose and KF quenching system for solution phase parallel synthesis

Amide 2

R

Yield (%)

Sulfonamide 3

R

Yield (%)

Urea 4

R

Yield (%)

a

Cyclopentyl (Sudrik et al. 2002)

98

a

Phenyl (José et al. 2011)

96

a

3-Cyano phenyl

98

b

t-Butyl (Martínez-Asencio et al. 2011a)

99

b

p-Tolyl (Gao et al. 2005)

99

b

1-Naphthyl

99

c

4-Fluro-phenyl (Mamat et al. 2011)

99

c

4-Fluro-phenyl (Ramunno et al. 2012)

97

c

4-Fluro phenyl

97

d

Cyclopropyl (Yang and Shi 2005)

94

d

4-Chlorophenyl (Ramunno et al. 2012)

98

d

2-Trifluromethyl-phenyl

98

e

Cyclohexyl (Saito et al. 2008)

98

e

4-Trifluromethoxy phenyl (Shi et al. 2009)

94

e

2-Methoxy-phenyl

97

f

n-Butyl (Dermer and King 1943)

97

f

4-Methoxy phenyl (Martínez-Asencio et al. 2011b)

99

f

Phenyl

99

g

2-Furyl (Gernigon et al. 2012)

99

g

2,4-Dichloro phenyl

98

g

4-Cyano phenyl

92

h

4-Nitro phenyl (Bahrami et al. 2010)

92

h

3,4-Dichloro phenyl

97

h

4-Triflurometh -oxy phenyl

94

i

4-Methoxy-phenyl (Kokare et al. 2007)

99

   

i

2,5-Dimethoxyphenyl

99

j

2,4-Dichloro-phenyl (Richard Cremlyna et al. 1989)

95

      

k

Ethyl (Lee et al. 1999)

97

      

l

Phenyl (Nowrouzi and Jonaghani 2012)

99

     Â